5-Fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c]-[1, 4]benzodiazepin-10(11H)-ylcarbonyl)-3-chlorophenyl]benzamide (VPA-985): an orally active arginine vasopressin antagonist with selectivity for V2 receptors.

J Med Chem

Wyeth-Ayerst Research, Pearl River, New York 10965, and Wyeth-Ayerst Research, Princeton, New Jersey 08543-8000, USA.

Published: July 1998

Download full-text PDF	Source
http://dx.doi.org/10.1021/jm980179c	DOI Listing

Publication Analysis

5-fluoro-2-methyl-n-[4-5h-pyrrolo[21-c]-[1 4]benzodiazepin-1011h-ylcarbonyl-3-chlorophenyl]benzamide

4]benzodiazepin-1011h-ylcarbonyl-3-chlorophenyl]benzamide vpa-985

vpa-985 orally

orally active

active arginine

arginine vasopressin

vasopressin antagonist

antagonist selectivity

selectivity receptors

5-fluoro-2-methyl-n-[4-5h-pyrrolo[21-c]-[1

Enter search terms and have AI summaries delivered each week - change queries or unsubscribe any time!