A versatile and convenient procedure for the functional derivatization with carbon substituents at the 6-position of pyridoxal using a Grignard reaction upon a protected -isobutoxycarbony-loxypyridoxal chloride and Heck reactions with protected 6-vinylpyridoxal has been developed.
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| http://dx.doi.org/10.1055/s-2000-6228 | DOI Listing |
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