Provided herein are novel pyrrolopyrazine compounds as ERK5 inhibitors, pharmaceutical compositions, use of such compounds in treating cancer, and processes for preparing such compounds.
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| http://dx.doi.org/10.1021/acsmedchemlett.4c00580 | DOI Listing |
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Pyrrolopyrazine Compounds as ERK5 Inhibitors for Treating Cancer.
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Smith, Gambrell & Russell LLP, 1105 W. Peachtree Street NE, Suite 1000, Atlanta, Georgia30309, United States.
Provided herein are novel pyrrolopyrazine compounds as ERK5 inhibitors, pharmaceutical compositions, use of such compounds in treating cancer, and processes for preparing such compounds.
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