Regioselective Synthesis of Quercetin and Myricetin Derivatives.

Russ J Gen Chem

Medical Pharmaceutical Institute, Pyatigorsk Branch of Volgograd Medical State University, 357532 Pyatigorsk, Russia.

Published: March 2023

A regioselective method for the synthesis of esters of quercetin and myricetin at the hydroxy group in the position 3 was developed. As acids participating in the esterification reaction, 2-hydroxybenzoic (salicylic), 4-hydroxybenzoic, 2,6-dihydroxybenzoic, 3,4-dihydroxybenzoic (procatechuic), 3,4,5-trihydroxybenzoic (gallic) acids were used. A new series of quercetin and myricetin esters were obtained.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC10062247PMC
http://dx.doi.org/10.1134/S1070363223020032DOI Listing

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