Synthesis of fluorescently labeled pyrazole derivative induceing a triple response in seedlings.

J Pestic Sci

Institute of Plant and Food Science, Department of Biology, School of Life Sciences, Southern University of Science and Technology (SUSTech).

Published: November 2022

A fluorescent labeled pyrazole derivative with a dansyl moiety () was synthesized. Design of was carried out by using a dansyl moiety to substitute the naphthalene moiety of the parent compound (). At a concentration of 30 µM, displayed biological activity on inducing a triple response in seedlings. Compared with the non-chemical treated control, the hypocotyl length of -treated seedlings was reduced from approximately 9.2±0.7 mm to 2.4±0.2 mm. The length of the roots was reduced from 1.7±0.1 mm to 1.0±0.1 mm, and the curvature of the hook of seedlings increased from 60±16 degrees to 245±35 degrees. The maxim excitation wavelength and emission wavelength of were 350 and 535 nm, respectively. Data obtained fluorescent microscope analysis indicated that intensive fluorescent signals of were observed in the shoot of seedlings.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC9716048PMC
http://dx.doi.org/10.1584/jpestics.D22-006DOI Listing

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