An efficient method for the selective preparation of trifluoromethyl-substituted azepin-2-carboxylates and their phosphorous analogues has been developed via Cu(I)-catalyzed tandem amination/cyclization reaction of functionalized allenynes with primary and secondary amines.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC9416787PMC
http://dx.doi.org/10.3390/molecules27165195DOI Listing

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