Voltage activation, but not channel opening, is required for RY785 to access the central cavity of Kv2 channels, where it promotes voltage sensor deactivation to trap itself in place.
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|---|---|
| http://www.ncbi.nlm.nih.gov/pmc/articles/PMC9086499 | PMC |
| http://dx.doi.org/10.1085/jgp.202213181 | DOI Listing |
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