An electro-oxidative cyclization pathway in which hydrazones are selected as starting materials to generate amphiphiles by reacting with benzylamines and benzamides was reported. This strategy successfully prepared a series of 1,2,4-triazoles in satisfactory yields. Moreover, the use of cheap stainless steel as the anode, the feasibility to conduct the transformation as a one-pot reaction and the proof that scaling-up these reactions is possible make this transformation attractive for potential application in industry.
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| http://www.ncbi.nlm.nih.gov/pmc/articles/PMC8792120 | PMC |
| http://dx.doi.org/10.1002/open.202100268 | DOI Listing |
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