An efficient method to assemble diverse benzoxazoles/benzothiazoles in good yields was developed via oxidative cyclization with 2-aminothiophenols or 2-iodoanilines as raw materials. In this protocol, elemental sulfur was used as the effective oxidant and C atoms on the C═C double bond were introduced as a one-carbon donator.

Download full-text PDF

Source
http://dx.doi.org/10.1021/acs.joc.1c01357DOI Listing

Publication Analysis

Top Keywords

c═c double
8
double bond
8
one-carbon donator
8
elemental sulfur-promoted
4
sulfur-promoted benzoxazole/benzothiazole
4
benzoxazole/benzothiazole formation
4
formation c═c
4
bond one-carbon
4
donator efficient
4
efficient method
4

Similar Publications

Want AI Summaries of new PubMed Abstracts delivered to your In-box?

Enter search terms and have AI summaries delivered each week - change queries or unsubscribe any time!