An operationally simple, scalable, and chemoselective method for the direct phosphorylation of alcohols using a P(V)-approach based on the Ψ-reagent platform is disclosed. The method features a broad substrate scope of utility in both simple and complex settings and provides access to valuable phosphorylated alcohols that would be otherwise difficult to obtain.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC8733960PMC
http://dx.doi.org/10.1021/acs.orglett.1c02736DOI Listing

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