Synthesis of 1,1-Diboryl Alkenes Using the Boryl-Heck Reaction.

Org Lett

Department of Chemistry and Biochemistry, University of Delaware, Newark, Delaware 19716, United States.

Published: June 2021

The synthesis of 1,1-diboryl alkenes from terminal alkenes is reported. 1,1-Regioselective addition is observed for both conjugated and unconjugated alkenes, allowing for a single method to prepare a wide range of 1,1-diboryl alkenes.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC8217338PMC
http://dx.doi.org/10.1021/acs.orglett.1c01567DOI Listing

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