AI Article Synopsis

  • Bumped kinase inhibitors (BKIs), specifically BKI 1369, effectively target calcium-dependent protein kinase 1 (CDPK1) to combat Cystoisospora suis, which causes coccidiosis in piglets.
  • The study tested the effectiveness of BKI 1369 with less frequent dosing, finding that a single treatment two days post-infection significantly reduced the replication of the parasite and oocyst excretion in infected piglets.
  • Treated piglets showed marked health improvements, including increased weight gain and fewer days of diarrhea, suggesting that less frequent use of BKI 1369 is a viable treatment option without adverse effects.

Article Abstract

Bumped kinase inhibitors (BKIs) are a new class of antiprotozoal drugs that target calcium-dependent protein kinase 1 (CDPK1) in various apicomplexan parasites. A multiple dose regimen of BKI 1369 has been shown to be highly effective against Cystoisospora suis (syn. Isospora suis), the causative agent of neonatal porcine coccidiosis. However, multiple dosing may not be widely applicable in the field. The present study aimed to determine the efficacy of reduced treatment frequencies with BKI 1369 against porcine cystoisosporosis in vitro and in vivo. Pre-incubation of sporozoites with BKI 1369 completely failed to inhibit the infection in vitro unless treatment was prolonged post-infection. Notably, a single treatment of infected cell cultures 2 days post-infection (dpi) resulted in a significant reduction of merozoite replication. In an experimental infection model, treatment of suckling piglets experimentally infected with C. suis 2 and 4 dpi with 20 mg BKI 1369/kg body weight completely suppressed oocyst excretion. A single treatment on the day of infection or 2 dpi suppressed oocyst excretion in 50% and 82% of the piglets and reduced the quantitative excretion in those that shed oocysts by 95.2% and 98.4%, respectively. Moreover, a significant increase in body weight gain and reduced number of diarrhea days were observed in BKI 1369 treated piglets compared to the control piglets, irrespective of time points and frequencies of treatment. Given that reduced treatment frequencies with BKI 1369 are comparable in efficacy to repeated applications without any adverse effects, this could be considered as a practical therapeutic alternative against porcine cystoisosporosis.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC7442133PMC
http://dx.doi.org/10.1016/j.ijpddr.2020.08.005DOI Listing

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