A conformationally constrained short peptide designed to target a protein-protein interaction hotspot in HIV-1 reverse transcriptase (RT) disrupts p66-p51 interactions and paves the way to the development of novel RT dimerization inhibitors.
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|---|---|
| http://www.ncbi.nlm.nih.gov/pmc/articles/PMC7236230 | PMC |
| http://dx.doi.org/10.1021/acsmedchemlett.9b00623 | DOI Listing |
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