was identified as a good starting point for modification, leading to an efficient and bio-available inhibitor for the SARS coronavirus main proteinase (SARS-CoV M). Synthesis of intermediate and analogues proceeded via a highly diastereoselective indium-mediated allylation of α-aminoaldehydes.
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|---|---|
| http://www.ncbi.nlm.nih.gov/pmc/articles/PMC7119068 | PMC |
| http://dx.doi.org/10.1016/j.tetlet.2004.10.146 | DOI Listing |
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