A dearomative tandem spiro-cyclization reaction of -[(1-indol-3-yl)methyl]methacrylamide derivatives with sulfinate sodium in the presence of AgNO and KCO is reported, which produced sulfonylated spiro[indole-3,3'-pyrrolidines] in medium to excellent yields. The characteristics of this transformation contain good functional group tolerance and ease of operation.

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http://dx.doi.org/10.1021/acs.orglett.0c00158DOI Listing

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