, 6-(1-Indol-4-yl)-8-methoxy-1-methyl-4-[1,2,4]triazolo[4,3-][1,4]benzodiazepine-4-acetic acid methyl ester, has been synthesized on a near-gram scale in seven steps with notable improvements in the reported poor-yielding last two steps enabling this key chemical probe compound to be available for researchers.
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| http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6641879 | PMC |
| http://dx.doi.org/10.1021/acsomega.7b00780 | DOI Listing |
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