A new, concise synthesis of the CCR-5 receptor antagonist maraviroc (UK-427,857) from 3-phenyl-1-propanol has been completed in four steps featuring a site-selective C-H functionalization.
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|---|---|
| http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4477708 | PMC |
| http://dx.doi.org/10.1016/j.tetlet.2015.01.074 | DOI Listing |
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