This report describes the discovery of RAD140, a potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM). The characterization of RAD140 in several preclinical models of anabolic androgen action is also described.
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| http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4018048 | PMC |
| http://dx.doi.org/10.1021/ml1002508 | DOI Listing |
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