Copper-catalyzed Chan-Lam coupling between sulfonyl azides and boronic acids at room temperature.

Org Lett

Department of Chemistry and Nano Science, Ewha Womans University, Global Top 5 Program, Seoul 120-750, Korea.

Published: January 2014

A mild and efficient method for the synthesis of N-arylsulfonamides in the presence of 10 mol % of CuCl is demonstrated. The reaction proceeds readily at room temperature in an open flask using a variety of sulfonyl azides and boronic acids without any base, ligand, or additive.

Download full-text PDF

Source
http://dx.doi.org/10.1021/ol403717fDOI Listing

Publication Analysis

Top Keywords

sulfonyl azides
8
azides boronic
8
boronic acids
8
room temperature
8
copper-catalyzed chan-lam
4
chan-lam coupling
4
coupling sulfonyl
4
acids room
4
temperature mild
4
mild efficient
4

Similar Publications

Want AI Summaries of new PubMed Abstracts delivered to your In-box?

Enter search terms and have AI summaries delivered each week - change queries or unsubscribe any time!