Synthesis and anti-toxoplasmosis activity of 4-arylquinoline-2-carboxylate derivatives.

Org Biomol Chem

Department of Chemistry and Chemical Biology, McMaster University, Hamilton, Ontario, Canada L8S 4M1.

Published: January 2014

A one-step synthesis of 4-arylquinoline-2-carboxylates along with their antiprotozoal activity against the pathogenic parasite Toxoplasma gondii is reported. Mechanistic insights into the role of Lewis acid (silver triflate) versus Bronsted acid (triflic acid) catalysis are revealed clarifying aspects of the mechanism of the quinoline synthesis.

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http://dx.doi.org/10.1039/c3ob41539bDOI Listing

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