A concise pathway to synthesize a novel class of pyrido(2,3-d)pyrimidine-C-β-D-glycosides.

Carbohydr Res

Department of Organic Chemistry, University of Madras, Guindy Campus, Chennai 25, Tamil Nadu, India.

Published: March 2013

A concise pathway to synthesize a novel class of nine different pyrido(2,3-d)pyrimidine-C-β-d-glycosides is reported. Formation of Michael adduct as an intermediate followed by heterocyclization are the key steps and the products were characterized by different spectral studies. β-Anomeric forms of C-glycosides were assigned from 1H NMR spectroscopy.

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http://dx.doi.org/10.1016/j.carres.2012.11.013DOI Listing

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