Stereocontrolled access to optically-enriched oxabispidines.

Chem Commun (Camb)

Pharmaceutical Development, AstraZeneca R&D Charnwood, Bakewell Road, Loughborough LE11 5RH, UK.

Published: May 2012

A range of chiral, optically-enriched bicyclic oxabispidines were prepared from (S)-(-)-2,3-epoxypropylphthalimide using an efficient sequence featuring a stereocontrolled intramolecular Mannich reaction as the key transformation.

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http://dx.doi.org/10.1039/c2cc30761hDOI Listing

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