The synthesis, photophysical and biological characterization of a small library of fluorescent 5-HT(3) receptor ligands is described. Several of these novel granisetron conjugates have high quantum yields and show high affinity for the human 5-HT(3)AR.
Download full-text PDF |
Source |
|---|---|
| http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3277886 | PMC |
| http://dx.doi.org/10.1016/j.bmcl.2011.11.097 | DOI Listing |
Publication Analysis
Top Keywords
5-ht3 receptor
8
high-affinity fluorescent
4
fluorescent ligands
4
ligands 5-ht3
4
receptor synthesis
4
synthesis photophysical
4
photophysical biological
4
biological characterization
4
characterization small
4
small library
4
Similar Publications
Want AI Summaries of new PubMed Abstracts delivered to your In-box?
Enter search terms and have AI summaries delivered each week - change queries or unsubscribe any time!