The synthesis of 2-aminobenzoxazoles can be readily achieved by two versatile, one-pot procedures utilizing commercially available tetramethyl orthocarbonate or 1,1-dichlorodiphenoxymethane, an amine, and an optionally substituted 2-aminophenol. The reactions were conducted under mild conditions and provided 2-aminobenzoxazoles in modest to excellent yields. A variety of amines and substituted 2-aminophenols were used to investigate the scope of the reactions.
Download full-text PDF |
Source |
|---|---|
| http://dx.doi.org/10.1021/jo1017052 | DOI Listing |
Publication Analysis
Top Keywords
synthesis 2-aminobenzoxazoles
8
tetramethyl orthocarbonate
8
orthocarbonate 11-dichlorodiphenoxymethane
8
2-aminobenzoxazoles tetramethyl
4
11-dichlorodiphenoxymethane synthesis
4
2-aminobenzoxazoles achieved
4
achieved versatile
4
versatile one-pot
4
one-pot procedures
4
procedures utilizing
4
Similar Publications
Want AI Summaries of new PubMed Abstracts delivered to your In-box?
Enter search terms and have AI summaries delivered each week - change queries or unsubscribe any time!