A high-throughput screening campaign resulted in the discovery of a highly potent dual cannabinoid receptor 1 (CB1) and 2 (CB2) agonist. Following a thorough SAR exploration, a series of selective CB2 full agonists were identified.
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| http://dx.doi.org/10.1016/j.bmcl.2008.01.042 | DOI Listing |
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