A 1000-member uridinyl branched peptide library was synthesized on PS-DES support using IRORI technology. High-throughput screening of this library for anti-tuberculosis activity identified several members with a MIC(90) value of 12.5 microg/mL.
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| http://dx.doi.org/10.1016/j.bmcl.2007.09.097 | DOI Listing |
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