Binding affinities for a range of epibatidine isomers and analogues at the alpha4beta2 and alpha3beta4 nAChR subtypes are reported; compounds having similar N-N distances to epibatidine show similar, high potencies.
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| http://dx.doi.org/10.1016/j.bmcl.2006.08.049 | DOI Listing |
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