Benzo[b]thiophene-2-carboxamides and benzo[b]furan-2-carboxamides have been found to be antagonists on the human histamine-3-receptor, showing a Ki value of as low as 4 nM.
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| http://dx.doi.org/10.1016/j.bmcl.2006.03.074 | DOI Listing |
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