A novel series of tetracyclic indoles have been designed, synthesized and evaluated as androgen receptor (AR) ligands. Studies of structure-activity relationships (SARs) were investigated, which led to some compounds in this series as strong binders to androgen receptors.
Download full-text PDF |
Source |
|---|---|
| http://dx.doi.org/10.1016/j.bmcl.2006.03.047 | DOI Listing |
Publication Analysis
Top Keywords
androgen receptor
8
receptor ligands
8
discovery indole-containing
4
indole-containing tetracycles
4
tetracycles scaffold
4
scaffold androgen
4
ligands novel
4
novel series
4
series tetracyclic
4
tetracyclic indoles
4
Similar Publications
Want AI Summaries of new PubMed Abstracts delivered to your In-box?
Enter search terms and have AI summaries delivered each week - change queries or unsubscribe any time!