A concise and diversity-oriented strategy for the synthesis of benzofurans and indoles via Ugi and Diels-Alder reactions.

Kui Lu Tuoping Luo Zheng Xiang Zejin You Reza Fathi Jiahua Chen Zhen Yang

J Comb Chem

Key Laboratory of Bioorganic Chemistry and Molecular Engineering of Ministry of Education, College of Chemistry, State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Science, Peking University, Beijing, China.

Published: January 2006

A one-pot synthesis of diverse benzofurans and indoles from readily available starting materials was achieved via the sequential Ugi four-component reaction, intramolecular Diels-Alder reaction, and oxidative aromatization.

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http://dx.doi.org/10.1021/cc050099b	DOI Listing

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