The synthesis of NPTS, 6, a potent inhibitor of the type 1 glycine transporter (GlyT1) is described, as well as preparation of 6 in optically active and tritiated form for use as a radioligand for affinity displacement assay of GlyT1.
Download full-text PDF |
Source |
|---|---|
| http://dx.doi.org/10.1016/s0960-894x(03)00126-4 | DOI Listing |
Publication Analysis
Top Keywords
type glycine
8
glycine transporter
8
[3h]-r-npts radioligand
4
radioligand type
4
transporter synthesis
4
synthesis npts
4
npts potent
4
potent inhibitor
4
inhibitor type
4
transporter glyt1
4
Similar Publications
Want AI Summaries of new PubMed Abstracts delivered to your In-box?
Enter search terms and have AI summaries delivered each week - change queries or unsubscribe any time!