1-Aryl-substituted primary cyclopropylamines are conveniently prepared from aromatic nitriles and diethylzinc. The yields range from 40 to 56% for donor-substituted (five examples) to 62-82% for non- and acceptor-substituted substrates (nine examples).
Download full-text PDF |
Source |
|---|---|
| http://dx.doi.org/10.1021/ol034021k | DOI Listing |
Publication Analysis
Top Keywords
primary 1-arylcyclopropylamines
4
1-arylcyclopropylamines aryl
4
aryl cyanides
4
cyanides diethylzinc
4
diethylzinc titanium
4
titanium alkoxides
4
alkoxides 1-aryl-substituted
4
1-aryl-substituted primary
4
primary cyclopropylamines
4
cyclopropylamines conveniently
4
Similar Publications
Primary 1-arylcyclopropylamines from aryl cyanides with diethylzinc and titanium alkoxides.
Org Lett
March 2003
Institut für Organische Chemie der Georg-August-Universität Göttingen, Tammannstrasse 2, 37077 Göttingen, Germany.
1-Aryl-substituted primary cyclopropylamines are conveniently prepared from aromatic nitriles and diethylzinc. The yields range from 40 to 56% for donor-substituted (five examples) to 62-82% for non- and acceptor-substituted substrates (nine examples).
View Article and Find Full Text PDFWant AI Summaries of new PubMed Abstracts delivered to your In-box?
Enter search terms and have AI summaries delivered each week - change queries or unsubscribe any time!