Novel antifungal beta-amino acids: synthesis and activity against Candida albicans.

Bioorg Med Chem Lett

Medicinal Chemistry, Business Group Pharma, Bayer AG, D-42096 Wuppertal, Germany.

Published: February 2003

A series of novel beta-amino acids has been synthesized and tested for their in vitro antifungal activity against Candida albicans. A steep SAR was observed. beta-Amino acid 21 (BAY 10-8888/PLD-118) revealed the most favourable activity-tolerability profile and was selected for clinical studies as a novel antifungal for the oral treatment of yeast infections.

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http://dx.doi.org/10.1016/s0960-894x(02)00958-7DOI Listing

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