Cyclooxygenase-2 inhibitors: promise or peril?

Mediators Inflamm

The Camden Group, 19 Oak Park Drive, St. Louis, MO 63141, USA.

Published: October 2002

The discovery of two isoforms of the cyclooxygenase enzyme, COX-1 and COX-2, and the development of COX-2-specific inhibitors as anti-inflammatories and analgesics have offered great promise that the therapeutic benefits of NSAIDs could be optimized through inhibition of COX-2, while minimizing their adverse side effect profile associated with inhibition of COX-1. While COX-2 specific inhibitors have proven to be efficacious in a variety of inflammatory conditions, exposure of large numbers of patients to these drugs in postmarketing studies have uncovered potential safety concerns that raise questions about the benefit/risk ratio of COX-2-specific NSAIDs compared to conventional NSAIDs. This article reviews the efficacy and safety profiles of COX-2-specific inhibitors, comparing them with conventional NSDAIDs.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC1781678PMC
http://dx.doi.org/10.1080/09629350290000041DOI Listing

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