Substituted 3-(2-benzoxazyl)-benzimidazol-2-(1H)-ones: a new class of GABA(A) brain receptor ligands.

Bioorg Med Chem Lett

Neurogen Corporation, Branford, CT 06405, USA.

Published: December 2000

A novel class of potent benzodiazepine receptor (BZR) ligands has been designed and synthesized aided by molecular modeling of known benzodiazepine ligands such as CGS-8216 and the use of known pharmacophore models.

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http://dx.doi.org/10.1016/s0960-894x(00)00550-3DOI Listing

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