Determination of the relative and absolute stereochemistry of a potent and alpha1A-selective adrenoceptor antagonist.

Bioorg Med Chem Lett

Department of Chemistry, Synaptic Pharmaceutical Corporation, Paramus, NJ 07652, USA.

Published: December 2000

The binding affinities and selectivities of antagonists 1-4 for the alpha1A-adrenoceptor are dependent on the stereochemical orientation of the groups at the C-4 and C-5 positions of the oxazolidinone ring. The unambiguous assignment of the relative and absolute configurations of the diastereomers of SNAP 7915 (1) is reported.

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http://dx.doi.org/10.1016/s0960-894x(00)00524-2DOI Listing

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